Drugs (By Class) (Last Updated - 12/14/2005)
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ACE Inhibitors (ACEI's):
1) Lisinopril (Prinivil)
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Anti-Coagulants:
A) Direct Thrombin Inhibitors:
1) Argatroban
2) Bivalirudin (Angiomax)
3) Lepirudin (Refludan)
B) Endogenous (Natural) Anti-Coagulants:
1) Prostaglandin I-2 (PGI-2 or Prostacyclin)
2) Anti-Thrombin
3) Heparan Sulfate
4) Protein C
5) Tissue Factor Pathway Inhibitor (TFPI or Extrinsic Pathway Inhibitor)
6) Thrombin (IIa)
C) Glycosaminoglycan Anti-Coagulants:
1) Heparin
2) Danaparoid (Orgaran)
3) Heparan Sulfate
4) Dermatan Sulfate
5) Chondroitin Sulfate
D) In Vitro Anti-Coagulants:
1) Heparan Sulfate
2) Dermatan Sulfate
3) Chondroitin Sulfate
E) Low Molecular Weight Heparins (LMWH's):
1) Enoxaparin (Lovenox)
2) Dalteparin (Fragmin)
3) Ardeparin (Normiflo)
4) Tinzaparin (Innohep) --> not FDA-approved
5) Nadroparin (Fraxiparine) --> not FDA-approved
6) Reviparin (Clivarine) --> not FDA-approved
F) Oral Anti-Coagulants:
1) Warfarin (Coumadin)
2) Acenocoumarol (Sinthrome)
3) Anisindione (Miradon)
4) Brodifacoum
5) Bromadiolone
6) Chlorophacinone
7) Diphenandione
8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
9) Phenprocoumon (Marcumar)
G) Pregnancy Anti-Coagulants:
1) Heparin --> DOC for anti-coagulation in pregnancy
H) Vitamin K Antagonists:
1) Warfarin (Coumadin)
2) Acenocoumarol (Sinthrome)
3) Anisindione (Miradon)
4) Brodifacoum
5) Bromadiolone
6) Chlorophacinone
7) Diphenandione
8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
9) Phenprocoumon (Marcumar)
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Antidotes:
1) Protamine Sulfate --> heparin antidote
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Direct Thrombin Inhibitors:
1) Argatroban
2) Bivalirudin (Angiomax)
3) Lepirudin (Refludan)
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Endogenous (Natural) Anti-Coagulants:
1) Prostaglandin I-2 (PGI-2 or Prostacyclin)
2) Anti-Thrombin
3) Heparan Sulfate
4) Protein C
5) Tissue Factor Pathway Inhibitor (TFPI or Extrinsic Pathway Inhibitor)
6) Thrombin (IIa)
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Glycosaminoglycan Anti-Coagulants:
1) Heparin
2) Danaparoid (Orgaran)
3) Heparan Sulfate
4) Dermatan Sulfate
5) Chondroitin Sulfate
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HMG-CoA Reductase Inhibitors (Statins):
1) Lovastatin (Mevacor)
2) Simvastatin (Zocor)
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In Vitro Anti-Coagulants:
1) Heparan Sulfate
2) Dermatan Sulfate
3) Chondroitin Sulfate
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Low Molecular Weight Heparins (LMWH's):
1) Enoxaparin (Lovenox)
2) Dalteparin (Fragmin)
3) Ardeparin (Normiflo)
4) Tinzaparin (Innohep) --> not FDA-approved
5) Nadroparin (Fraxiparine) --> not FDA-approved
6) Reviparin (Clivarine) --> not FDA-approved
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Oral Anti-Coagulants:
1) Warfarin (Coumadin)
2) Acenocoumarol (Sinthrome)
3) Anisindione (Miradon)
4) Brodifacoum
5) Bromadiolone
6) Chlorophacinone
7) Diphenandione
8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
9) Phenprocoumon (Marcumar)
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Pregnancy Anti-Coagulants:
1) Heparin
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Rodenticides:
1) Bromadiolone
2) Brodifacoum
3) Diphenandione
4) Chlorophacinone
5) Phenindione (Dindevan or Pindione)
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Statins (HMG-CoA Reductase Inhibitors):
1) Lovastatin (Mevacor)
2) Simvastatin (Zocor)
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Thrombolytics:
1) t-PA (Tissue Plasminogen Activator)
2) Alteplase (Activase)
3) Anistreplase (Eminase)
4) Prourokinase (Saruplase) --> not FDA-approved
5) Reteplase (Retavase)
6) Streptokinase (Streptase) --> DOC
7) Urokinase (Abbokinase)
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Vitamin K Antagonists:
1) Warfarin (Coumadin)
2) Acenocoumarol (Sinthrome)
3) Anisindione (Miradon)
4) Brodifacoum
5) Bromadiolone
6) Chlorophacinone
7) Diphenandione
8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
9) Phenprocoumon (Marcumar)
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