Drugs (By Class) (Last Updated - 12/14/2005)

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ACE Inhibitors (ACEI's):

     1) Lisinopril (Prinivil)

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Anti-Coagulants:

     A) Direct Thrombin Inhibitors:

          1) Argatroban
          2) Bivalirudin (Angiomax)
          3) Lepirudin (Refludan)

     B) Endogenous (Natural) Anti-Coagulants:

          1) Prostaglandin I-2 (PGI-2 or Prostacyclin)
          2) Anti-Thrombin
          3) Heparan Sulfate
          4) Protein C
          5) Tissue Factor Pathway Inhibitor (TFPI or Extrinsic Pathway Inhibitor)
          6) Thrombin (IIa)

     C) Glycosaminoglycan Anti-Coagulants:

          1) Heparin
          2) Danaparoid (Orgaran)
          3) Heparan Sulfate
          4) Dermatan Sulfate
          5) Chondroitin Sulfate

     D) In Vitro Anti-Coagulants:

          1) Heparan Sulfate
          2) Dermatan Sulfate
          3) Chondroitin Sulfate

     E) Low Molecular Weight Heparins (LMWH's):

          1) Enoxaparin (Lovenox)
          2) Dalteparin (Fragmin)
          3) Ardeparin (Normiflo)
          4) Tinzaparin (Innohep) --> not FDA-approved
          5) Nadroparin (Fraxiparine) --> not FDA-approved
          6) Reviparin (Clivarine) --> not FDA-approved

     F) Oral Anti-Coagulants:

          1) Warfarin (Coumadin)
          2) Acenocoumarol (Sinthrome)
          3) Anisindione (Miradon)
          4) Brodifacoum
          5) Bromadiolone
          6) Chlorophacinone
          7) Diphenandione
          8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
          9) Phenprocoumon (Marcumar)

     G) Pregnancy Anti-Coagulants:

          1) Heparin --> DOC for anti-coagulation in pregnancy

     H) Vitamin K Antagonists:

          1) Warfarin (Coumadin)
          2) Acenocoumarol (Sinthrome)
          3) Anisindione (Miradon)
          4) Brodifacoum
          5) Bromadiolone
          6) Chlorophacinone
          7) Diphenandione
          8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
          9) Phenprocoumon (Marcumar)

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Antidotes:

     1) Protamine Sulfate --> heparin antidote

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Direct Thrombin Inhibitors:

     1) Argatroban
     2) Bivalirudin (Angiomax)
     3) Lepirudin (Refludan)

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Endogenous (Natural) Anti-Coagulants:

     1) Prostaglandin I-2 (PGI-2 or Prostacyclin)
     2) Anti-Thrombin
     3) Heparan Sulfate
     4) Protein C
     5) Tissue Factor Pathway Inhibitor (TFPI or Extrinsic Pathway Inhibitor)
     6) Thrombin (IIa)

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Glycosaminoglycan Anti-Coagulants:

     1) Heparin
     2) Danaparoid (Orgaran)
     3) Heparan Sulfate
     4) Dermatan Sulfate
     5) Chondroitin Sulfate

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HMG-CoA Reductase Inhibitors (Statins):

     1) Lovastatin (Mevacor)
     2) Simvastatin (Zocor)

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In Vitro Anti-Coagulants:

     1) Heparan Sulfate
     2) Dermatan Sulfate
     3) Chondroitin Sulfate

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Low Molecular Weight Heparins (LMWH's):

     1) Enoxaparin (Lovenox)
     2) Dalteparin (Fragmin)
     3) Ardeparin (Normiflo)
     4) Tinzaparin (Innohep) --> not FDA-approved
     5) Nadroparin (Fraxiparine) --> not FDA-approved
     6) Reviparin (Clivarine) --> not FDA-approved

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Oral Anti-Coagulants:

     1) Warfarin (Coumadin)
     2) Acenocoumarol (Sinthrome)
     3) Anisindione (Miradon)
     4) Brodifacoum
     5) Bromadiolone
     6) Chlorophacinone
     7) Diphenandione
     8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
     9) Phenprocoumon (Marcumar)

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Pregnancy Anti-Coagulants:

     1) Heparin

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Rodenticides:

     1) Bromadiolone
     2) Brodifacoum
     3) Diphenandione
     4) Chlorophacinone
     5) Phenindione (Dindevan or Pindione)

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Statins (HMG-CoA Reductase Inhibitors):

     1) Lovastatin (Mevacor)
     2) Simvastatin (Zocor)

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Thrombolytics:

     1) t-PA (Tissue Plasminogen Activator)
     2) Alteplase (Activase)
     3) Anistreplase (Eminase)
     4) Prourokinase (Saruplase) --> not FDA-approved
     5) Reteplase (Retavase)
     6) Streptokinase (Streptase) --> DOC
     7) Urokinase (Abbokinase)

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Vitamin K Antagonists:

     1) Warfarin (Coumadin)
     2) Acenocoumarol (Sinthrome)
     3) Anisindione (Miradon)
     4) Brodifacoum
     5) Bromadiolone
     6) Chlorophacinone
     7) Diphenandione
     8) Phenindione (Dindevan or Pindione) --> no longer recommended for use by the FDA
     9) Phenprocoumon (Marcumar)

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